A series of arylidene thiosemicarbazides have been prepared by a new method, which was titled as transalkylidation. This method is an effective, fast, green and clean method. The mechanism of this reaction has been discussed.
Mohamed A. El-Atawy +3 more
doaj +1 more source
Co-infection of malaria and tuberculosis, although not thoroughly investigated, has been noted. With the increasing prevalence of tuberculosis in the African region, wherein malaria is endemic, it is intuitive to suggest that the probability of co ...
Richard M. Beteck +6 more
doaj +1 more source
Decoding Urease Inhibition: A Comprehensive Review of Inhibitor Scaffolds
Representative functional groups known for urease inhibition are reviewed within diverse scaffolds using structure–activity analyses to identify features associated with high inhibitory activity. Urease is a metalloenzyme produced by a wide range of organisms and plays a critical role in nitrogen microbial metabolism by catalyzing the hydrolysis of ...
Nuno Martinho, Natália Aniceto
wiley +1 more source
Synthesis, Characterization, Crystal Structures and Urease Inhibition of Thiosemicarbazones
Thiosemicarbazones are biological active compounds. Six new thiosemicarbazones were prepared and structurally characterized by elemental analysis, 1H NMR and IR spectra, as well as single crystal X-ray diffraction.
Ling-Wei Xue, Qiao-Ru Liu, Yong-Jun Han
doaj +1 more source
ABSTRACT Background and Aims The escalation of chronic wounds necessitates advanced therapeutic strategies beyond current interventions. Hydrogel dressings, particularly injectable hydrogels, offer promising solutions due to their water absorption capacity, structural resilience, and ease of application.
Mohammad Ebrahim Astaneh +5 more
wiley +1 more source
Background and purpose: This study aimed to evaluate the cytotoxicity of synthesized thiosemicarbazone derivatives, particularly on biomarkers associated with ferroptosis.
Yasaman Shadmani +4 more
doaj +1 more source
Synthesis and structural characterization of a disulphide-bridged tetranuclear palladium(II) complex derived from 3,5-diacetyl 1,2,4-triazole bis(4-ethylthiosemicarbazone) [PDF]
NOTICE: this is the author’s version of a work that was accepted for publication in Inorganic Chemistry Communications. Changes resulting from the publishing process, such as peer review, editing, corrections, structural formatting, and other quality ...
Matesanz, Ana I. +2 more
core +2 more sources
Cyclopalladated Complexes With Functionalized Diphosphanes as Promising Antifungal Scaffolds
Invasive fungal infections, especially those caused by Candida spp., have been classified as a serious global threat. The emergence of species intrinsically resistant to current drugs, along with the increase in acquired resistance, places significant pressure on the need to develop novel and more effective antifungal agents.
Cláudia Malta-Luís +13 more
wiley +1 more source
Mono- és bisz(acil)hidrazonok átalakulásai: Gyűrűs N,O,S-acetálok/ketálok szintézise. = Transformations of mono- and bis(acyl)hydrazones: Synthesis of cyclic N,O,S-acetals/ketals. [PDF]
Aldehid- és keton-tioszemikarbazonokat állítottunk elő, melyeket acilezési körülmények között 3-acil-1,3,4-tiadiazolinokká ciklizáltunk. A 2-monoszubsztituált heterogyűrűs vegyületek oxidáló, illetve dehidrogénező szerek [kálium permanganát és a most ...
Somogyi, László
core
New bioactive 2,6-diacetylpyridine bis(p-chlorophenylthiosemicarbazone) ligand and its Pd(II) and Pt(II) complexes: Synthesis, characterization, cytotoxic activity and DNA binding ability [PDF]
NOTICE: this is the author’s version of a work that was accepted for publication in Journal of Inorganic Biochemistry. Changes resulting from the publishing process, such as peer review, editing, corrections, structural formatting, and other quality ...
Hernández, Carolina +2 more
core +2 more sources

