Electrochemical TEMPO-Catalyzed Oxidative Ugi-Type Reaction [PDF]
ACS Organic & Inorganic Au, 2021 Oxidative isocyanide-based multicomponent reactions (oxidative IMCRs) are very useful tools for the rapid construction of molecular diversity starting from readily available and stable substrates. Despite all their benefits, such multicomponent reactions are underdeveloped and strictly limited to 3-component processes.
Na Pan +4 more
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Direct polymerization of levulinic acid via Ugi multicomponent reaction [PDF]
, 2016 A robust, direct and efficient approach has been developed for the utilization of levulinic acid (LevA) as a building block in the synthesis of polyamides.
Manuel Hartweg, C. Remzi Becer
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Unimolecular Exciplexes by Ugi Four-Component Reaction [PDF]
Frontiers in Chemistry, 2019 Exciplex or excited complex emission is an excited state process, arising from considerable charge transfer of an excited energy donor to an acceptor, which can be identified by the occurrence of a redshifted emission band that is absent in the ...
Maria Ochs +3 more
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Rh(III)-Catalyzed C-2 Alkylation of Indoles followed by a Post-Synthetic Modification via the Ugi Reaction. [PDF]
ChemistryOpen, 2023 Januário MAP +3 more
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Diastereoselective Ugi reaction of chiral 1,3-aminoalcohols derived from an organocatalytic Mannich reaction [PDF]
Beilstein Journal of Organic Chemistry, 2016 Enantiomerically pure β-aminoalcohols, produced through an organocatalytic Mannich reaction, were subjected to an Ugi multicomponent reaction under classical or Lewis acid-promoted conditions with diastereoselectivities ranging from moderate to good ...
Samantha Caputo +5 more
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Silver(I) triflate-catalyzed post-Ugi synthesis of pyrazolodiazepines [PDF]
Beilstein Journal of Organic ChemistryA silver(I) triflate-catalyzed post-Ugi assembly of novel pyrazolo[1,5-a][1,4]diazepine scaffolds is reported offering high yields (up to 98%) under mild conditions.
Muhammad Hasan +6 more
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Synthesis of various N-heterocycles using the four-component Ugi reaction
ACS Combinatorial Science, 2019 Ugi four-component reactions (U-4CRs) are widely recognized as being highly efficient for the synthesis of pseudopeptides. However, the products of these reactions are not so interesting as drug candidates because they are not conformationally restricted enough for a potent interaction with biological targets.
Majid M. Heravı, Leyla Mohammadkhani
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Propargyl Amines: Versatile Building Blocks in Post‐Ugi Transformations
ChemistryOpen, 2023 The Ugi reaction, a multicomponent reaction, allows diversity‐oriented synthesis Its importance is recognized by an exponential increase in the publications utilizing the post‐Ugi transformations as a strategy to build complex molecules via simple and ...
Rinkal B. Bhoraniya, Dr. Sachin G. Modha
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Turn-Induction in Peptides Incorporating Novel Cyrene-Derived α,α-Disubstituted Amino Acid. [PDF]
J Pept SciNovel chiral cyrene‐derived Cyr residues were incorporated into peptides. The α,α‐disubstituted amino acid residue was introduced using the Ugi reaction. X‐ray crystallographic analysis of R‐ and S‐Cyr residues indicated preference to adopt left‐ and right‐handed α‐helical conformations, respectively.
Bhowal KB, Hitti R, Lubell WD.
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Recent Progress on Post-Ugi Reaction [PDF]
Chinese Journal of Organic Chemistry, 2017 Xiuming Li, Xueshun Jia, Liang Yin
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