Results 121 to 130 of about 14,756 (172)

Navigating the complexities of drug development for metallo-β-lactamase inhibitors. [PDF]

RSC Med Chem
Reddy N, Balieiro AM, Silva JRA, Gouws CA, Mutshembele A, Arvidsson PI, Kruger HG, Govender T, Naicker T.   +8 more
europepmc   +1 more source

Penicillin-Binding Protein Occupancy Dataset for 18 β-Lactams and 4 β-Lactamase Inhibitors in Neisseria gonorrhoeae. [PDF]

Microbiol Spectr, 2023
López-Argüello S, Montaner M, Mármol-Salvador A, Velázquez-Escudero A, Docobo-Pérez F, Oliver A, Moya B.   +6 more
europepmc   +1 more source

Restoring ceftolozane susceptibility: a role for diazabicyclooctane β-lactamase inhibitors? [PDF]

Antimicrob Agents Chemother
Dorazio AJ, Kline EG, Squires KM, Pogue JM, Van Tyne D, Shields RK.   +5 more
europepmc   +1 more source

Role of β-lactamase inhibitors on cefiderocol activity against carbapenem-resistant Acinetobacter species. [PDF]

Int J Antimicrob Agents, 2023
Mezcord V, Wong O, Pasteran F, Corso A, Tolmasky ME, Bonomo RA, Ramirez MS.   +6 more
europepmc   +1 more source

Harder than Metal: Challenging Antimicrobial Resistance with Metallo-β-lactamase Inhibitors. [PDF]

J Med Chem
De Falco A, Alfano AI, Cutarella L, Mori M, Brindisi M.   +4 more
europepmc   +1 more source

Challenges of Carbapenem-Resistant <i>Enterobacteriaceae</i> in the Development of New β-Lactamase Inhibitors and Antibiotics. [PDF]

Antibiotics (Basel)
Leroux P, Bornet C, Bolla JM, Cohen A.
europepmc   +1 more source

Sustainable Joullié-Ugi and Continuous Flow Implementation Led to Novel Captopril-Inspired Broad-Spectrum Metallo-β-Lactamase Inhibitors. [PDF]

J Med Chem
Alfano AI, Pelliccia S, Barone S, Cutarella L, Cancade SMI, Baia V, Cassese E, Russomanno P, Messano N, Frank D, Weizel L, Rotter MJ, Brunst S, Wichelhaus TA, Proschak E, Tedesco D, Mori M, Docquier JD, Summa V, Brindisi M.   +19 more
europepmc   +1 more source

Efflux Pump (QacA, QacB, and QacC) and β-Lactamase Inhibitors? An Evaluation of 1,8-Naphthyridines against Staphylococcus aureus Strains. [PDF]

Molecules, 2023
Oliveira-Tintino CDM, Tintino SR, Justino de Araújo AC, Dos Santos Barbosa CR, Ramos Freitas P, Araújo Neto JB, Begnini IM, Rebelo RA, Silva LED, Mireski SL, Nasato MC, Krautler MIL, Barreto HM, Ribeiro-Filho J, de Menezes IRA, Coutinho HDM.   +15 more
europepmc   +1 more source

Discovery of Boronic Acids-Based β-Lactamase Inhibitors Through In Situ Click Chemistry. [PDF]

Int J Mol Sci
Santi N, Piccirilli A, Corsini F, Taracila MA, Perilli M, Bonomo RA, Fini F, Prati F, Caselli E.   +8 more
europepmc   +1 more source

<i>In vitro</i> activity of cefiderocol against <i>Pseudomonas aeruginosa</i> demonstrating evolved resistance to novel β-lactam/β-lactamase inhibitors. [PDF]

JAC Antimicrob Resist, 2023
Shields RK, Kline EG, Squires KM, Van Tyne D, Doi Y.   +4 more
europepmc   +1 more source