Identification and characterization of antibacterial compound(s) of cockroaches (Periplaneta americana) [PDF]
, 2017 Infectious diseases remain a significant threat to human health, contributing to more than 17 million deaths, annually. With the worsening trends of drug resistance, there is a need for newer and more powerful antimicrobial agents.
A Brüning +215 more
core +1 more source
Synthesis of substituted 1, 2, 4-triazole derivatives by Microwave irradiation [PDF]
IOSR Journal of Applied Chemistry, 2013 Various substituted Triazole-Thiol containing different functional group have been synthesized by microwave method. The title product 1-((3H-indol-2-ylamino) methyl)-4-phenyl-4, 5-dihydro-1H-1, 2, 4- triazole-3-thiol is synthesized by using amino benzothiazole.
Ashish Asrondkar +2 more
openaire +1 more source
Microwave-assisted Eco-Friendly Synthesis and Antimicrobial Evaluation of Aryl-Triazole-1,3,4-Thiadiazols [PDF]
, 2017 Due to the growing awareness about environmental pollution and environmental legislation, recent years have witnessed a phenomenal increase in the application of microwave irradiation (MW) in organic synthesis.
Dwivedi, Smriti, Jaiswal, Shalini
core +2 more sources
Synthesis and Biological Activities of Some 1,2,4-Triazole Derivatives: A Review [PDF]
, 2022 This review is about 1,2,4-triazoles include their synthesis; their physio-chemical properties, SAR, reactions, derivatives. Finally, their biological activities with a demonstrated showing different requirements to achieve different ...
Ayad Kareem Khan +2 more
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Ultrasound promoted green synthesis of benzofuran substituted thiazolo[3,2-b][1,2,4]triazoles
Green Processing and Synthesis, 2017 A highly efficient, eco-friendly and one-pot synthesis of benzofuran substituted thiazolo[3,2-b][1,2,4]triazoles was developed involving the reaction of 2-acetyl benzofurans and 5-mercapto-3-(4-chlorophenyl)-1,2,4triazole in the presence of molecular ...
Kumar Surender, Sharma Dinesh Kumar
doaj +1 more source
Microwave assisted metal-free approach to access 1,2,3-triazoles through multicomponent synthesis
Current Research in Green and Sustainable Chemistry, 2020 The work illustrates multicomponent reaction of aldehydes, nitroalkanes and sodium azide for the metal-free synthesis of N-unsubstituted-1,2,3-triazoles using anthranilic acid as an organocatalyst under microwave irradiation. This is the first ever green
Anirban Garg +2 more
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Chemical properties of amino- and thio-derivatives of 1,2,4-triazoles
Aktualʹnì Pitannâ Farmacevtičnoï ì Medičnoï Nauki ta Praktiki, 2015 Aim. A number of references of the last ten years have been carefully studied with bibliosemantic method to compile information on the participation of 1,2,4-triazoles in chemical reactions. Introduction of new domestic drugs intopractice, which could
A. G. Kaplaushenko
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HUBUNGAN KUANTITATIF STRUKTUR DAN AKTIVITAS SENYAWA TURUNAN BENZIMIDAZOL TERTAUTKAN 1,2,3-TRIAZOL SEBAGAI INHIBITOR ENZIM α-GLUKOSIDASE [PDF]
, 2023 ABSTRAK Penemuan obat diabetes mellitus sedang banyak dilakukan akibat meningkatnya angka penderita diabetes mellitus. Peneliti menemukan penghambatan terhadap enzim α-glukosidase berperan penting dalam mencegah diabetes komplikasi dan mengontrol gula ...
Nurkholidah, Intan +2 more
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Novel 4-thiazolidinone derivatives as agonists of benzodiazepine receptors [PDF]
A new series of 4-chloro-N-(2-(substitutedphenyl)-4-oxothiazolidin-3-yl)-2-phenoxybenzamide derivatives were designed, synthesized and biologically evaluated as anticonvulsant agents.
Almasirad, Ali +7 more
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Фармацевтичний журнал, 2018 Chemistry of heterocyclic compounds is one of the most popular sector in organic chemistry. Scientists allocate among them a class of derivatives of 1,2,4-triazole.
I. I. Aksyonova-Seliuk +2 more
doaj +1 more source