Results 101 to 110 of about 37,211,421 (159)

GABA(A) receptor phospho-dependent modulation is regulated by phospholipase C-related inactive protein type 1, a novel protein phosphatase 1 anchoring protein [PDF]

, 2004
GABA(A) receptors are critical in controlling neuronal activity. Here, we examined the role for phospholipase C-related inactive protein type 1 (PRIP-1), which binds and inactivates protein phosphatase 1alpha (PP1alpha) in facilitating GABA(A) receptor ...
Kanematsu, T, Terunuma, M, Jovanovic, JN, Jang, IS, Kittler, JT, Akaike, N, Nakayama, KI, Ryu, SH, Moss, SJ, Ha, SH, Hirata, M   +10 more
core  

Mutational and computational characterization of transmembrane domains in the fungal G protein-coupled pheromone receptors STE2 and Mam2 [PDF]

G protein-coupled receptors (GPCRs) comprise the largest family of cell-surface receptors involved in sensing a multitude of ligands and are consequently attractive pharmacological targets.
Nilsson Lock, Gun Antonia Evelina
core  

Overlapping and opposing functions of G protein-coupled receptor kinase 2 (GRK2) and GRK5 during heart development. [PDF]

J Biol Chem, 2014
Philipp M, Berger IM, Just S, Caron MG.
europepmc   +1 more source

G Protein-Coupled Receptor Kinase 2 (GRK2) and 5 (GRK5) Exhibit Selective Phosphorylation of the Neurotensin Receptor in Vitro. [PDF]

Biochemistry, 2015
Inagaki S, Ghirlando R, Vishnivetskiy SA, Homan KT, White JF, Tesmer JJ, Gurevich VV, Grisshammer R.   +7 more
europepmc   +1 more source

Pharmacological inhibition of G protein-coupled receptor kinase 2 (GRK2) by paroxetine attenuates acetaminophen-induced hepatotoxicity. [PDF]

Korean J Physiol Pharmacol
Yang D, Moon HW, Kim JW, Kim B.
europepmc   +1 more source

Recent advances in the development of GRK2 inhibitors: blocking the interaction of GRK2 with its partners. [PDF]

Acta Pharmacol Sin
Han CC, Guo HZ, Guo FY, Tan HZ, Sun HZ, Gu JT, Zuo SJ, Wang WK, Ma Y, Wei W.   +9 more
europepmc   +1 more source

G protein-coupled receptor kinase 3 regulates CCR7 signaling, trafficking, and T cell responses to CCL19 and CCL21. [PDF]

J Biol Chem
Sanchez A, Cardona CI, Kaiser B, Bill CA, Miller ME, Bassuk DW, Wagener BM, Brissette MA, Ibanez D, Llano M, Bill CA, Vines CM.   +11 more
europepmc   +1 more source

G protein-coupled receptor kinase 3 couples atypical chemokine receptor 4 independent of G proteins. [PDF]

Mol Pharmacol
Lamme TD, Sánchez Arroyo IB, Smit MJ, Schafer CT.   +3 more
europepmc   +1 more source

Molecular Mechanisms of Electroacupuncture-Induced Spinal Microglial Reprogramming in Neuropathic Pain: A Systematic Search-Narrative Review. [PDF]

Brain Sci
Teoh BK, Nguyen TTH, Peddanna K, Quach TVB, Lin JG, Chen YH.   +5 more
europepmc   +1 more source

G-protein regulatory network governs receptor internalization dynamics. [PDF]

Proc Natl Acad Sci U S A
Rowe JB, Pandey S, Mayer RA, Ludlam WG, Drube J, Inoue A, Hoffmann C, Martemyanov KA.   +7 more
europepmc   +1 more source