Results 111 to 120 of about 11,559 (254)

SEMI-EXPERIMENTAL EQUILIBRIUM STRUCTURE OF 1,3-OXAZOLE FROM MANY ISOTOPOLOGUES [PDF]

, 2023
Brian J. Esselman, Robert J. McMahon
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Design, synthesis, and pharmacological evaluation of N-(3-carbamoyl-1H-pyrazol-4-yl)-1,3-oxazole-4-carboxamide derivatives as interleukin-1 receptor-associated kinase 4 inhibitors with reduced potential for cytochrome P450 1A2 induction

, 2023
Hiroshi Inami, Tsuyoshi Mizutani, Junko Watanabe, Hisashi Hayashida, Tomonori Ito, Takeshi Terasawa, Toru Kontani, Hiroaki Yamagishi, Hiroyuki Usuda, Naohiro Aoyama, Emiko Imamura, Takeshi Ishikawa   +11 more
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Synthesis and biological evaluation of 4-(1H-imidazol-2-yl)-2-(pyrimidin-5-yl)oxazoles as potent anticancer agents

Results in Chemistry
A new series of aryl derivatives of 4-(1H-imidazol-2-yl)-2-(pyrimidin-5-yl)oxazoles 11a–j were synthesised and their structures were characterized by analytical techniques.
Divya Komirishetti, Vasantha Mittapelli
doaj   +1 more source

ONE-POT SYNTHESES OF 2-(1H-BENZO[d]OXAZOLE-2-YL)-N-ARYLBENZAMIDES BY SELF-CATALYSIS [PDF]

, 2019
V. Ramesh, G. Purna Chander Rao, D. Ramachandran, A. Kalyan Chakravarthy   +3 more
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Targeting the Hsp90 interactome using in silico polypharmacology approaches [PDF]

, 2013
In recent years, polypharmacology has gained popularity in drug discovery. [1] Especially for complex diseases such as cancer, the ability of a drug to bind to and interfere with multiple targets provides new opportunities for therapeutic intervention ...
Anighoro, Andrew, Bajorath, J., Heikamp, K., Rastelli, Giulio, Stumpfe, D.   +4 more
core  

Theoretical design of new bridge-ring insensitive high energy compounds by selected normal Diels-Alder reactions between NH2-substituted oxazoles and NO2/NF2/NHNO2-substituted ethylenes/acetylenes

, 2020
Qiong Wu, Qinnan Hu, Mingquan Li, Ze-wu Zhang, Weihua Zhu   +4 more
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Synthesis and pharmacological trials of new phosphorylated oxazole derivatives antihypertensive properties

, 2020
Iryna Nizhenkovska, Kateryna V. Matskevych, A. V. Golovchenko, Oksana I. Golovchenko   +3 more
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Alkynyl Thioethers in Gold‐Catalyzed Annulations To Form Oxazoles [PDF]

, 2017
Raju Jannapu Reddy, Matthew P. Ball‐Jones, Paul Davies   +2 more
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Synthesis and biological evaluation of chalcone derivatives of oxazole-pyrimidines as anticancer agents

Results in Chemistry
We have developed a new library of chalcone derivatives of oxazole-pyrimidines (16a-j) and their structures were confirmed by analytical data. Further, in vitro anticancer activity of the newly prepared compounds 16a-j was assessed against a panel of ...
Divya Komirishetti, Tasqeeruddin Syed, Vasantha Mittapelli   +2 more
doaj   +1 more source

Synthesis and HDAC inhibitory activity of isosteric thiazoline-oxazole largazole analogs

, 2013
Jennifer M. Guerra-Bubb, Albert A. Bowers, William Smith, Ronald M. Paranal, Guillermina Estiú, Olaf Wiest, James E. Bradner, Robert M. Williams   +7 more
openalex   +1 more source