α-Ketoglutaric acid in Ugi reactions and Ugi/aza-Wittig tandem reactions. [PDF]
Honcharov VO +6 more
europepmc +1 more source
Targeted Treatment of Cancer by Using Conjugate Compounds with Poly(ADP-ribose) Polymerase (PARP) Inhibitors. [PDF]
Zhou X, Liang SH.
europepmc +1 more source
Natural and Synthetic Peptides as Alternatives to Antibiotics in Intestinal Infections-A Review. [PDF]
Stepanyan L +9 more
europepmc +1 more source
Concise Synthesis of Optically Active Cyclopropane β-Amino Acid Derivatives via Olefination of Cyclopropanone Surrogates. [PDF]
Jung M, Lindsay VNG.
europepmc +1 more source
Functionalised peptidomimetic metallohelices [PDF]
Chapter 1 introduces small host-defence peptides in cancer therapy. The main mechanisms proposed in their interactions with membranes and intracellular targets are discussed. The biologically relevant peptide mimetics are also reviewed.\ud \ud Chapter 2 describes the synthesis and characterisation of alkyne derivatives of metallohelices.
openaire
Poly(ethylene Glycol)-Based Peptidomimetics (Pegtides) of Antimicrobial Peptides. [PDF]
Shine C +13 more
europepmc +1 more source
AlphaFold-Guided Discovery of an Overlapping MYC/Miz-1 Interface Enables Peptidomimetic Disruption of MYC/MAX. [PDF]
Ellenbroek BD +2 more
europepmc +1 more source
Synthesis, Antimicrobial Activity, and Tyrosinase Inhibition by Multifunctional 3,4-Dihydroxy-Phenyl Peptidomimetics. [PDF]
Wavhal DS +4 more
europepmc +1 more source
A Polyproline Type II Peptidomimetic Disrupts a Grb2 SH3C Domain Protein-Protein Interaction Implicated in Breast Cancer. [PDF]
Luccarelli J +4 more
europepmc +1 more source

