Synthesis of some Nitro-substituted 1,3,4-Oxadiazoles, 1,3,4-Thiadiazoles and 1,2,4-Triazoles as Antiamebic Agents [PDF]
, 1989 Post-Graduate Department of Chemistry, University of Jammu, Jammu-180 004 Manuscript received 20 May 1987, revised 15 November 1988, accepted 14 December 1988 Some 2-(\(\beta\)-arylethyl)-5-phenylamino-1,3,4-oxadiazoles, 2-(\(\beta\)-arylethyl)-5 ...
T. C. LANGER +2 more
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Synthesis and Antimicrobial Activity of Some New 1,3,4-Thiadiazole Derivatives
Molecules, 2012 New series of 1,3,4-thiadiazoles have been prepared via reaction of 1,3,4-thiadiazolenaminones 1 with N-phenyl 2-oxopropanehydrazonoyl chloride (2) in dioxane in the presence of triethylamine.
Mohamed R. Abdel Aziz +2 more
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Synthesis, Characterization, and Antimicrobial Properties of New 1,3,4‐Thiadiazoles Derived from Azo Dyes [PDF]
, 2019 Some new 1,3,4‐thiadiazoles derived from azo dyes were synthesized. Two different synthesis methods were used for these compounds: Esters pertaining to the azo dyes were converted into 1,3,4‐thiadiazoles, or benzothiazole ester derivatives were converted
Gür, Mahmut, Mahmut Gür
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Synthesis of some substituted 1,3,4-oxadiazoles, thiadiazoles and 1,2,4-triazoles [PDF]
مجلة التربية والعلم, 2009 In this paper the synthesis of some substituted 1,3,4-oxadiazoles, 1,3,4-thiadiazoles and 1,2,4-triazoles is reported. Ethyl methacrylate was treated with hydrazine hydrate in ethanol to give the corresponding hydrazide (1).
Shereen R. Mohamed
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Journal of Enzyme Inhibition and Medicinal Chemistry, 2023 A novel series of 12 antipyrine derivatives containing 1,3,4-oxadiazoles (4a-d), 1,3,4-thiadiazoles (6a-d), and pyrimidines (8a-d), was preparedand assessed for its potential in vitro COX-2 inhibitors.
Mohammad M. Al-Sanea +11 more
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Synthesis and Cytotoxic Activity of New 1,3,4-Thiadiazole Thioglycosides and 1,2,3-Triazolyl-1,3,4-Thiadiazole N-glycosides [PDF]
Molecules, 2019 New 1,3,4-thiadiazole thioglycosides linked to substituted arylidine systems were synthesized via glycosylation of the prepared 1,3,4-thiadiazole thiol compounds. Click strategy was also used for the synthesis of new 1,3,4-thiadiazole and 1,2,3-triazole hybrid glycosides by reaction of the acetylenic derivatives with different glycosyl azids followed ...
Fahad M. Alminderej +4 more
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Synthesis and antiproliferative studies of 5-aryl-2-(3-thienylamino)-1,3,4- thiadiazoles [PDF]
, 2014 A series of 5-aryl-2-(3-thienylamino)-1,3,4-thiadiazoles 3a-m were synthesized in good yields in two steps starting from thiophen-3- isothiocyanates.
Gadais, Charlène +4 more
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SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF NEW N-ETHYL-N-METHYL BENZENE SULFONAMIDE DERIVATIVES [PDF]
Al-Azhar Journal of Pharmaceutical Sciences, 2014 This article describes the synthesis of some novel sulfonamide having the biologically active hydrazones 1,3,4-thiadiazoles and 4-oxothiazolidines moieties 2-4, 7 and 10-13 respectively. Starting with 4-acetyl-N-ethyl-N-methyl benzene sulfonamide (
Ahmed El-Morsy
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Greener and rapid access to bio-active heterocycles: one-pot solvent-free synthesis of 1,3,4-oxadiazoles and 1,3,4-thiadiazoles [PDF]
, 2008 A novel one-pot solvent-free synthesis of 1,3,4-oxadiazoles and 1,3,4-thiadiazoles by condensation of acid hydrazide and triethyl orthoalkanates under microwave irradiations is reported.
Polshettiwar, Vivek, Varma, Rajender S.
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Synthesis of 1,3,4-Thiadiazole Derivatives and Their Anticancer Evaluation
International Journal of Molecular Sciences, 2023 Thiadiazole derivatives have garnered significant attention in the field of medicinal chemistry due to their diverse pharmacological activities, including anticancer properties. This article presents the synthesis of a series of thiadiazole derivatives and investigates their chemical characterization and potential anticancer effects on various cell ...
Camelia Elena Stecoza +8 more
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