Results 61 to 70 of about 12,547 (208)
Molecules, 2010 New 5-(2-thienyl)-1,2,4-triazoles and 5-(2-thienyl)-1,3,4-oxadiazoles namely, N-[3-mercapto-5-(2-thienyl)-1,2,4-triazol-4-yl]-N'-arylthioureas 4a–e, 2-arylamino-5-(2-thienyl)-1,2,4-triazolo[3,4-b][1,3,4]thiadiazoles 5a–e, 3-arylaminomethyl-5-(2-thienyl ...
Mohamed A. Al-Omar
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Electrophilic Iodination of Heterocyclic Compounds. Recent Advances 2008–2025: Part II
European Journal of Organic Chemistry, Volume 29, Issue 22, 9 June 2026.Electrophilic iodination using molecular iodine and iodide sources represents an efficient approach for accessing valuable iodinated organic compounds. This review highlights recent advances in the iodination of heterocyclic compounds from 2008 to 2025, emphasizing the role of heteroaryl iodides as important synthetic intermediates for biologically ...
Njomza Ajvazi, Stojan Stavber
wiley +1 more source
Preparation and evaluation of some 1,3,4-thiadiazoles as diuretic agents [PDF]
, 2004 184-188Sixteen newer 2-(substituted acetamido)-5-aryl- 1,3,4-thiadiazoles have been prepared and screened for LD50 and diuretic activity. A few of the compounds namely 4a1, 4a2 and 4c3 shows diuretic activity comparable with the standard drug ...
P. Mishra +3 more
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Designed Lewis Acid–Base Passivation for High Performance Perovskite Solar Cells
Advanced Functional Materials, Volume 36, Issue 51, 25 June 2026.ABSTRACT Silicon's high cost and long energy payback time remain major barriers to the global expansion of solar power. In contrast, metal–halide perovskites offer abundant, solution‐processable absorbers, and have achieved efficiencies of 25%–30%, positioning them as strong competitors to silicon.
Afna Manaf +4 more
wiley +1 more source
A Selective Phenyl Azo Acetate Substrate for Enhanced Carbonic Anhydrase Functional Analysis
Analytical Science Advances, Volume 7, Issue 1, June 2026.ABSTRACT Carbon dioxide (CO2) sequestration is a key strategy for mitigating climate change, and biocatalytic approaches offer sustainable, cost‐effective alternatives to chemical and physical methods. Carbonic anhydrases (CAs) efficiently catalyse the reversible hydration of CO2 to bicarbonate, yet their large‐scale application is constrained by ...
Justinas Babinskas, Inga Matijošytė
wiley +1 more source
Cumhuriyet Science Journal, 2018 1,3,4-Thiadiazoles have a variety of biologicalactivities depending on their substituents. This study aims to investigatethe in vitro antioxidant properties of 1R,2R-1,2-bis- (5- (4-hydroxynaphthalen-1-ylazo) - [1,3,4] thiadiazol-2-yl) -ethane- 1,2-diole
Akif Evren Parlak, Pelin Koparır
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Journal of Taibah University for Science, 2022 One of the worst diseases, cancer claims millions of lives each year throughout the world, necessitating the creation of novel treatments. In this study, we designed a novel series of 1,3,4-thiadiazoles through the reaction of 2-(4-methyl-2-(2-(1 ...
Ghadah F. Aljohani +6 more
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Medicinal Insights Into FLT3 Inhibitors as Anticancer Agents: Current Status and Future Direction
Archiv der Pharmazie, Volume 359, Issue 6, June 2026.Structure–activity relationship of FMS‐like tyrosine kinase 3 (FLT3) as potent anti‐cancer agents supported by biological evaluation, in silico and clinical trial studies. ABSTRACT FMS‐like tyrosine kinase 3 (FLT3) is a receptor tyrosine kinase (RTK) important for hematopoietic stem cell proliferation, differentiation, and survival.
Ankush Kumar +4 more
wiley +1 more source
Synthesis and in vitro antibacterial activity evaluation of coumarin-1,3,4-thiadiazoles hybrids [PDF]
Purpose: Hybridization of two or more potent pharmacophores into a single molecule is one of the current strategies to synthesize compounds with improved pharmacological activity.
Asrat, Ergena
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An efficient synthesis of styryl 1,3,4-thiadiazoles using Lawesson’s reagent and Propylphosphonic anhydride-precursors for bis heterocycles [PDF]
, 2014 The compounds styryl 1,3,4-thiadiazoles were prepared adopting one and two step methodologies to optimize the yield of the products. The two-step methodology via benzohydrazide followed by treatment with Lawesson’s reagent in the presence of ...
Padmavathi, Venkatapuram +3 more
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