Results 91 to 100 of about 629 (164)

Synthesis, bioactivity, and molecular docking studies: novel arylpiperazine derivatives as potential new-resistant AR antagonists. [PDF]

Front Chem
Jiang H, Chen H, Wang Y, Xu H, Chen H.
europepmc   +1 more source

Bioisosteric Replacement of Amides with 1,2,3-Triazoles Improves Dopamine D4 Receptor Ligand Pharmacokinetics. [PDF]

ACS Pharmacol Transl Sci
Alkhatib M, Jakobs FM, Hanson JN, Nilson AN, Moritz AE, Li T, Faibille AB, Bourn LA, Ramdhan PA, Ricchezza J, Jordan S, Panasis D, Nguyen N, Kasarla N, Wang B, Garcia SS, Saez J, Paule J, Lee CB, Rais R, Slusher BS, Sibley DR, Li C, Keck TM, Boateng CA.   +24 more
europepmc   +1 more source

Green synthesis of 1,3,5-triazine derivatives using a sonochemical protocol. [PDF]

Ultrason Sonochem
Kułaga D, Drabczyk AK, Zaręba P, Jaśkowska J, Chrzan J, Ewa Greber K, Ciura K, Plażuk D, Wielgus E.   +8 more
europepmc   +1 more source

Hybrid design reveals a dopamine D3R ligand with promising in vitro ADME properties. [PDF]

Bioorg Chem
Namballa HK, Dorogan M, Patra S, Gudipally A, Xie L, Xie L, Harding WW.   +6 more
europepmc   +1 more source

CXCR3 inhibitors for therapeutic interventions: current status and perspectives. [PDF]

Front Pharmacol
Huo R, Jiang Y, Zhang L, Du S, Zhou D.
europepmc   +1 more source

Identification of oxyresveratrol, a food-as-medicine substrate, as a novel EPI that targets the RND efflux pumps of <i>Serratia surfactantfaciens</i> sp. nov. YD25^T. [PDF]

Microbiol Spectr
Liu F, Wei X, Lou Y, Wang Y, Zhang D, Cao B, Su C, Sun Y, Li Z.   +8 more
europepmc   +1 more source

Preclinical Pharmacokinetics and Pharmacodynamics of Antibiotic Adjuvants. [PDF]

ACS Infect Dis
Pham VT, De Oliveira DMP, Kuo A, Walker MJ, Smith MT.   +4 more
europepmc   +1 more source

A Systematic Review of Inverse Agonism at Adrenoceptor Subtypes. [PDF]

Cells, 2020
Michel MC, Michel-Reher MB, Hein P.
europepmc   +1 more source

Regulation, structure, and activity of the <i>Pseudomonas aeruginosa</i> MexXY efflux system. [PDF]

Antimicrob Agents Chemother
Kavanaugh LG, Hinrichsen ME, Dunham CM, Conn GL.   +3 more
europepmc   +1 more source

Synthesis and evaluation of arylpiperazines derivatives of 3,5-dioxo-(2H,4H)-1,2,4-triazine as 5-HT1AR ligands. [PDF]

Bioorg Med Chem Lett, 2014
Kumar JSD, Majo VJ, Prabhakaran J, Mann JJ.   +3 more
europepmc   +1 more source