Results 111 to 120 of about 44,050 (359)

A facile synthesis and anticancer activity of some novel thiazoles carrying 1,3,4-thiadiazole moiety

open access: yesChemistry Central Journal, 2017
BackgroundThiazoles and 1,3,4-thiadiazoles have been reported to possess various pharmacological activities.ResultsA novel series of thiazoles carrying 1,3,4-thiadiazole core were designed and prepared via the reaction of the 2-(4-methyl-2-phenylthiazole-
Sobhi M. Gomha   +4 more
semanticscholar   +1 more source

Design and Synthesis of Triazole‐Based p‐tert‐Butylcalix[4]Arene Conjugates and Evaluation of Their Antimicrobial, Antibiofilm, and Anti‐Quorum‐Sensing Activities

open access: yesBiotechnology and Applied Biochemistry, EarlyView.
ABSTRACT Macrocyclic calix[n]arenes have many applications, with diverse structures that can easily be functionalized either on upper or lower rims, mostly to impart solubility and improve biological activities. In this study, triazole‐based p‐tert‐butylcalix[4]arene conjugates (AT10a and AT10b) and their p‐tert‐butylphenol analogs (AT10b and AT11b ...
Alfred Ngenge Tamfu   +2 more
wiley   +1 more source

Oxazole and thiazole analogs of sulindac for cancer prevention [PDF]

open access: yes, 2018
Aim: Experimental and epidemiological studies and clinical trials suggest that nonsteroidal anti-inflammatory drugs possess antitumor potential. Sulindac, a widely used nonsteroidal anti-inflammatory drug, can prevent adenomatous colorectal polyps and ...
Connelly, Michele C.   +4 more
core   +2 more sources

The Relationship Between Aldose Reductase and Isoxazole Derivatives: An In Vitro and In Silico Approach to Its Correlation With Diabetic Conditions

open access: yesBiotechnology and Applied Biochemistry, EarlyView.
ABSTRACT Diabetes mellitus (DM), which can result in a number of problems such as cataracts, neuropathy, retinopathy, nephropathy, and several cardiovascular illnesses, continues to be a growing issue despite major advancements in treatment approaches.
Ahmet Esat Göner, Hatice Esra Duran
wiley   +1 more source

Thiopeptide antibiotics: retrospective and recent advances [PDF]

open access: yes, 2014
Thiopeptides, or thiazolyl peptides, are a relatively new family of antibiotics that already counts with more than one hundred different entities.
Albericio Palomera, Fernando   +2 more
core   +3 more sources

UPLC‐ESI‐QTOF‐MS/MS Profiling, Antioxidant, and Cytotoxicity Potentials of Marrubium vulgare L. Extracts: Experimental Analysis and Computational Validation

open access: yesChemistry &Biodiversity, EarlyView.
ABSTRACT Plant extracts are emerging as valuable options for food additives and therapeutic treatments. This study evaluated the phytochemical profile, antioxidant activity, and cytotoxicity of aerial parts of Marrubium vulgare L. crude extract (MVCE) and its subfractions.
Ines El Mannoubi   +8 more
wiley   +1 more source

RESEARCH REGARDING THE POTENTIAL ACTIVITY OF SOME HETEROCYCLIC COMPOUNDS ON PLANTS GROWTH AND DEVELOPMENT

open access: yesScientific Study & Research: Chemistry & Chemical Engineering, Biotechnology, Food Industry, 2017
It is well known that growth and morphogenesis of plant tissue cultures can be improved by small amounts of some organic compounds. Heterocyclic compounds such as chromanones and thiazoles derivatives, valuable because of their potential biological ...
OANA-IRINA PATRICIU   +6 more
doaj  

N-Propargylamines: versatile building blocks in the construction of thiazole cores

open access: yesBeilstein Journal of Organic Chemistry, 2017
Thiazoles and their hydrogenated analogues are not only key structural units in a wide variety of natural products but they also constitute important building blocks in medicinal chemistry.
S. Arshadi   +4 more
doaj   +1 more source

Functionalization of Silicon Surface by Thiadiazole Molecule : a DFT Study

open access: yes, 2018
The first principles density functional theory (DFT) calculations have been used to investigate the atomic and electronic properties of thiadiazole adsorption on the Si(001) surface.
Kaderoglu, Cagil
core   +1 more source

Safety evaluation of substituted thiophenes used as flavoring ingredients. [PDF]

open access: yes, 2016
This publication is the second in a series by the Expert Panel of the Flavor and Extract Manufacturers Association summarizing the conclusions of its third systematic re-evaluation of the safety of flavorings previously considered to be generally ...
Bastaki, M   +11 more
core   +1 more source

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