Results 11 to 20 of about 45,916 (341)
Thiazole Ring—A Biologically Active Scaffold [PDF]
Molecules, 2021 Background: Thiazole is a good pharmacophore nucleus due to its various pharmaceutical applications. Its derivatives have a wide range of biological activities such as antioxidant, analgesic, and antimicrobial including antibacterial, antifungal ...
Anthi Petrou +2 more
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Reactions of acryl thioamides with iminoiodinanes as a one-step synthesis of N-sulfonyl-2,3-dihydro-1,2-thiazoles [PDF]
Beilstein Journal of Organic ChemistryA one-step method has been developed for the preparation of 2,3-dihydro-2-sulfonyl-3,4,5-substituted 1,2-thiazoles by the reaction of acryl thioamides and iminoiodinanes.
Vladimir G. Ilkin +7 more
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3-Phenylpropanal and citral in the multicomponent synthesis of novel thiopyrano[2,3-d]thiazoles
Results in Chemistry, 2022 A 3-phenylpropanal and citral were studied in the multicomponent reaction with the isorhodanine and maleimides (EDDA catalyst) with the aim of the novel thiopyrano[2,3-d]thiazoles synthesis.
Andrii Lozynskyi +6 more
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Photochemical permutation of thiazoles, isothiazoles and other azoles. [PDF]
NatureThiazoles and isothiazoles are privileged motifs in drug and agrochemical discovery1,2. The synthesis of these derivatives is generally approached, designed and developed on a case-by-case basis. Sometimes, the lack of robust synthesis methods to a given
Roure B +12 more
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Thiazolylcyanocyclopropanes: Novel Donor–Acceptor Cyclopropanes for Accessing Thiazole-Containing Targets [PDF]
MoleculesDonor–acceptor (D–A) cyclopropanes are important precursors in the synthesis of complex molecules due to their bidentate character and high reactivity.
Emanuèl Bruno Savini +5 more
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Scientific Reports, 2023 Microbial infections are currently a widespread disease in hospitals and community health centres and are a major cause of death worldwide. In pursuit of searching new antimicrobial agents, coumarin linked to thiazoles, pyridines and pyrazoles have been ...
Mariam T. Sayed +2 more
semanticscholar +1 more source
Pyridin-2-ylthiazolothiazoles – Synthesis and photophysical properties
Results in Chemistry, 2021 Thiazolo[5,4-d]thiazoles are valuable materials for a range of technical and biological applications. They are used as chemosensors, electroluminescent materials, organic light-emitting diodes (OLEDs), in solar cells, in live-cell imaging, etc., and for ...
Ana F.R. Cerqueira +3 more
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Molecules, 2021 Rapidly growing antimicrobial resistance among clinically important bacterial and fungal pathogens accounts for high morbidity and mortality worldwide.
Dovilė Malūkaitė +6 more
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Indian Journal of Pharmaceutical Education and Research, 2022 Thiazole or 1,3-thiazole is a distinct heterocyclic compound which incorporates sulphur and nitrogen atoms. It is a vital framework present in numerous pharmacologically active compounds, be it of natural origin or of synthetic nature.
Shivkant Sharma +4 more
semanticscholar +1 more source
Acta Chimica Slovenica, 2021 One of the best ways to design new biocidal agents is synthesizing hybrid molecules by combining two or more bioactive moieties in a single molecular scaffold.
Mohamed Salem +8 more
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