Results 11 to 20 of about 44,050 (359)
Thiazole Derivatives of Aminopropanes. [PDF]
Torsten Ekstrand+2 more
openalex +3 more sources
In this article, we applied ultrasonic irradiation as an ecofriendly, green, efficient approach for the synthesis of a new 1,3-thiazoles and 1,3,4-thiadiazines under solvent-free conditions.
Sara N. Shabaan+3 more
doaj +1 more source
Identification of 2-Aminothiazole-4-Carboxylate Derivatives Active against Mycobacterium tuberculosis H37Rv and the β-Ketoacyl-ACP Synthase mtFabH [PDF]
Background Tuberculosis (TB) is a disease which kills two million people every year and infects approximately over one-third of the world's population.
Abbott, G+13 more
core +5 more sources
Thiazoles, their benzofused systems, and thiazolidinone derivatives are widely recognized as nuclei of great value for obtaining molecules with various biological activities, including analgesic, anti-inflammatory, anti-HIV, antidiabetic, antitumor, and ...
S. Cascioferro+6 more
semanticscholar +1 more source
Review of the synthesis and biological activity of thiazoles
This study covers the literature documents available on the chemistry of preparation of thiazoles. Additionally, we cover the biological activities of certain thiazoles.
Sukinah H. Ali, A. R. Sayed
semanticscholar +1 more source
Biosynthesis of the Thiamin-Thiazole in Eukaryotes: Identification of a Thiazole Tautomer Intermediate [PDF]
Thiamin thiazole biosynthesis in eukaryotes is still not completely understood. In this report, a late intermediate, tightly bound to the active site of the Saccharomyces cerevisiae thiazole synthase, was identified as an adenylated thiazole tautomer. The reactivity of this unusual compound was evaluated.
Abhishek Chatterjee+4 more
openaire +3 more sources
The Panel on Food additives and Flavourings (FAF) was requested to evaluate the flavouring substances 2,4‐dimethyl‐3‐thiazoline [FL‐no: 15.060] and 2‐isobutyl‐3‐thiazoline [FL‐no: 15.119] in Flavouring Group Evaluation 21 revision 6 (FGE.21Rev6).
EFSA Panel on Food Additives and Flavourings (FAF)+25 more
doaj +1 more source
Several new thiazole derivatives linked pyrazole and/or pyridine rings were synthesized based on the versatile precursor 2-(5-acetyl-4-methyl-3-phenylthiazol-2(3H)-ylidene)acetonitrile (1). The synthesized derivatives were optimized using DFT approach in order to inspect the configurations and energies of the HOMO-LUMO orbitals.
Abrar Bayazeed+7 more
openaire +2 more sources
One-Pot Synthesis of Novel Thiazoles as Potential Anti-Cancer Agents
Background Thiazole and thiosemicarbazone derivatives are known to have potential anticancer activity with a mechanism of action related to inhibition of matrix metallo-proteinases, kinases and anti-apoptotic BCL2 family proteins. Materials and Methods A
A. R. Sayed+6 more
semanticscholar +1 more source