Novel hybrid thiazoles, bis-thiazoles linked to azo-sulfamethoxazole: Synthesis, docking, and antimicrobial activity [PDF]
HeliyonThe reaction of sulfamethoxazolehydrazonoyl chloride with thiosemicarbazones, bis-thiosemicarbazones, or 4-amino-3-mercapto-1,2,4-triazole in dioxane in the presence of triethylamine as a basic catalyst at reflux resulted in the regioselective synthesis ...
Mostafa E. Salem +7 more
doaj +2 more sources
Identification of 2-Aminothiazole-4-Carboxylate Derivatives Active against Mycobacterium tuberculosis H37Rv and the β-Ketoacyl-ACP Synthase mtFabH [PDF]
, 2009 Background Tuberculosis (TB) is a disease which kills two million people every year and infects approximately over one-third of the world's population.
Abbott, G +13 more
core +3 more sources
Iridium-Catalyzed Silylation of Five-Membered Heteroarenes: High Sterically Derived Selectivity from a Pyridyl-Imidazoline Ligand. [PDF]
, 2020 The steric effects of substituents on five-membered rings are less pronounced than those on six-membered rings because of the difference in bond angles. Thus, the regioselectivities of reactions of five-membered heteroarenes that occur with selectivities
Hartwig, John F +3 more
core +1 more source
Journal of Saudi Chemical Society, 2015 A rapid synthesis of hydrazinyl thiazoles under solvent and catalyst free condition is reported within 30 s. A series of aryl ketones/4-benzoyl pyridine thiosemicarbazone, thiosemicarbazide and α-haloketones were used.
D. Chinnaraja, R. Rajalakshmi
doaj +1 more source
Cyclic peptide production using a macrocyclase with enhanced substrate promiscuity and relaxed recognition determinants [PDF]
, 2017 This project was supported by grants from the ERC (no. 339367, MJ), BBSRC IBCatalyst (no. BB/M028526/1, MJ, WEH), BBSRC FoF (no. BB/M013669/1, MJ, WEH), IBioIC Exemplar (no. 2014-2-4, MJ, WEH), an AstraZeneca studentship (MJ, WEH, LT, KR), the Academy of
Alexandru-Crivac, Cristina N. +16 more
core +1 more source
Structure of the cyanobactin oxidase ThcOx from Cyanothece sp. PCC 7425, the first structure to be solved at Diamond Light Source beamline I23 by means of S-SAD [PDF]
, 2016 Acknowledgements We thank Diamond Light Source for providing access to beamline I23. We also thank Thomas Sorensen and his staff for access to and support on beamline I02.
Bent, Andrew F +8 more
core +1 more source
A Facile Synthesis of 2,4-Disubstituted Thiazoles Using MnO2
Molecules, 2009 Structurally diverse thiazoles with electron-donating and electron-withdrawing groups were conveniently synthesized through manganese dioxide (MnO2) oxidation of the corresponding thiazolines.
Bin Fu +4 more
doaj +1 more source
Applied Sciences, 2021 The reaction of 2-(1-(2-(2-(4-methoxybenzylidene)hydrazinyl)-4-methylthiazol-5-yl)ethylidene)hydrazinecarbothioamide with a range of hydrazonoyl chlorides and α-halo-compounds yielded three new series of thiazole derivatives.
Laila A. Al-Mutabagani +7 more
doaj +1 more source
Effet inhibiteur à la longues chaînes et de dérivés thiazolés sur la corrosion du laiton Amirauté.optimale des petites stations d'épuration à boues activées [PDF]
, 1995 Dans cette étude, des mesures électrochimiques ont été réalisées pour caractériser le comportement du laiton Amirauté dans une solution de chlorure de sodium 0,5 M en l'absence d'inhibiteur et en présence d'un mélange d'amines à longue chaîne et de ...
Blériot, P. +3 more
core +1 more source
3-Phenylpropanal and citral in the multicomponent synthesis of novel thiopyrano[2,3-d]thiazoles
Results in Chemistry, 2022 A 3-phenylpropanal and citral were studied in the multicomponent reaction with the isorhodanine and maleimides (EDDA catalyst) with the aim of the novel thiopyrano[2,3-d]thiazoles synthesis.
Andrii Lozynskyi +6 more
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